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[61] Like numerous other cardiotoxic drugs, methadone blocks the hERG K+ channel. The two enantiomers of methadone inhibit hERG channels with distinctive potency. Dextromethadone, and that is a lot less potent as an opioid, is a lot more powerful at blocking the hERG channel with an IC50 of ~twelve μM. Levomethadone incorporates a lower affinity,